Bahaa El-Dien M. El-Gendy|Publications

Benha University

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Dr. Bahaa El-Dien M. El-Gendy :: Publications:

Research Fields

Organic Synthesis

Nuclear Magnetic Resonance (NMR)

Medicinal Chemistry

Natural Products

Nuclear Hormone Receptors

Drug Discovery

Computational Chemistry

Number of publications is 32

Title

1-Structure-based design and synthesis of conformationally constrained derivatives of methyl-piperidinopyrazole (MPP) with estrogen receptor (ER) antagonist activity

2-Identification of Novel Mitochondrial Pyruvate Carrier Inhibitors by Homology Modeling and Pharmacophore-Based Virtual Screening

Abstract' | Full paper

3-Ligand-based design, synthesis, computational insights, and in vitro studies of novel N-(5-Nitrothiazol-2-yl)-carboxamido derivatives as potent inhibitors of SARS-CoV-2 main protease

4-Synthesis and Evaluation of Troponoids as a New Class of Antibiotics

5-Identification of novel small molecule inhibitors against the NS3/4A protease of hepatitis C virus genotype 4a

6-Development of novel liver X receptor modulators based on a 1, 2, 4-triazole scaffold

7-Identification of 4-isopropyl–thiotropolone as a novel anti-microbial: regioselective synthesis, NMR characterization, and biological evaluation

8-Recent Advances in the Medicinal Chemistry of Liver X Receptors

9-P450 3A-Catalyzed O-Dealkylation of Lapatinib Induces Mitochondrial Stress and Activates Nrf2

10-Investigation of adsorption and inhibition effects of some novel anil compounds towards mild steel in H 2 SO 4 solution: Electrochemical and theoretical quantum studies

11-Broad anti-tumor activity of a small molecule that selectively targets the warburg effect and lipogenesis

12-Stereoselective Synthesis, Structural and Spectroscopic Study of 4, 5, 11-Triazatricyclo [6.2. 1.0* 2, 6*] Undec-5-ene

13-Antibacterial activity of diketopiperazines isolated from a marine fungus using t-butoxycarbonyl group as a simple tool for purification

14-Pyrrolizines: Promising scaffolds for anticancer drugs

15-Pharmacological targeting of the mammalian clock regulates sleep architecture and emotional behaviour

16-Regioselective synthesis, stereochemical structure, spectroscopic characterization and geometry optimization of dispiro[3H-indole-3,2′-pyrrolidine-3′,3″-piperidines]

17-A Liver-Selective LXR Inverse Agonist That Suppresses Hepatic Steatosis

18-Small molecule amides as potent ROR-γ selective modulators

19-α-Substitution Effects on the Ease of S→N-Acyl Transfer in Aminothioesters

20-Synthesis of Benzoxazines, Quinazolines and 4H-Benzo[e][1,3]thiazine by ANRORC Rearrangements of 1,2,4-Oxadiazoles

21-Synthesis of chiral α-amino acid-derived 1H-1,2,4-triazoles and 1,2,4-triazines

22-Efficient microwave-assisted synthesis of aminoxy acid conjugates

23-Cyclohexanol analogues are positive modulators of GABAA receptor currents and act as general anaesthetics in vivo

24-Synthesis and photochemistry of pH-sensitive GFP chromophore analogs

25-NMR Study of the Tautomeric Behavior of N-(α-Aminoalkyl)tetrazoles

26-Conformational equilibria and barriers to rotation in some novel nitroso derivatives of indolizines and 3- and 5-azaindolizines – an NMR and molecular modeling study

27-Tautomerism in drug discovery

28-1H, 13C, and 15N NMR spectra of some pyridazine derivatives

29-Tautomerism of guanidines studied by 15N NMR: 2-hydrazono-3-phenylquinazolin-4 (3H)-ones and related compounds

30-Selective Synthesis and Structural Elucidation of S-Acyl- and N-Acylcysteines

31-(α -Aminoacyl)amino-substituted heterocycles and related compounds

32-Benzotriazole-mediated alkoxyalkylation and acyloxyalkylation

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